1qiv
HEADER    CALCIUM-BINDING PROTEIN                 17-JUN-99   1QIV              
TITLE     CALMODULIN COMPLEXED WITH N-(3,3,-DIPHENYLPROPYL)-N'-[1-R-(           
TITLE    2 3,4-BIS-BUTOXYPHENYL)-ETHYL]-PROPYLENEDIAMINE (DPD), 1:2             
TITLE    3 COMPLEX                                                              
COMPND    MOL_ID: 1;                                                            
COMPND   2 MOLECULE: CALMODULIN;                                                
COMPND   3 CHAIN: A                                                             
SOURCE    MOL_ID: 1;                                                            
SOURCE   2 ORGANISM_SCIENTIFIC: BOS TAURUS;                                     
SOURCE   3 ORGANISM_COMMON: BOVINE;                                             
SOURCE   4 ORGAN: BRAIN;                                                        
SOURCE   5 CELLULAR_LOCATION: CYTOPLASM                                         
KEYWDS    CALCIUM-BINDING PROTEIN                                               
EXPDTA    X-RAY DIFFRACTION                                                     
AUTHOR    V.HARMAT,Z.S.BOCSKEI,B.G.VERTESSY,G.NARAY-SZABO,J.OVADI               
REVDAT   1   28-MAR-00 1QIV    0                                                
JRNL        AUTH   V.HARMAT,Z.S.BOCSKEI,G.NARAY-SZABO,I.BATA,                   
JRNL        AUTH 2 A.S.CSUTOR,I.HERMECZ,P.ARANYI,B.SZABO,K.LILIOM,              
JRNL        AUTH 3 B.G.VERTESSY,J.OVADI                                         
JRNL        TITL   A NEW POTENT CALMODULIN ANTAGONIST WITH                      
JRNL        TITL 2 ARYLALKYLAMINE STRUCTURE: CRYSTALLOGRAPHIC,                  
JRNL        TITL 3 SPECTROSCOPIC AND FUNCTIONAL STUDIES                         
JRNL        REF    J.MOL.BIOL.                   V. 297   747 2000              
JRNL        REFN   ASTM JMOBAK  UK ISSN 0022-2836                               
REMARK   1                                                                      
REMARK   1 REFERENCE 1                                                          
REMARK   1  AUTH   B.G.VERTESSY,V.HARMAT,Z.S.BOCSKEI,G.NARAY-SZABO,             
REMARK   1  AUTH 2 F.OROSZ,J.OVADI                                              
REMARK   1  TITL   SIMULTANEOUS BINDING OF DRUGS WITH DIFFERENT                 
REMARK   1  TITL 2 CHEMICAL STRUCTURES TO CA 2+ CALMODULIN:                     
REMARK   1  TITL 3 CRYSTALLOGRAPHIC AND SPECTROSCOPIC STUDIES                   
REMARK   1  REF    BIOCHEMISTRY                  V.  37 15300 1998              
REMARK   1  REFN   ASTM BICHAW  US ISSN 0006-2960                               
REMARK   1 REFERENCE 2                                                          
REMARK   1  AUTH   B.G.VERTESSY,Z.S.BOCSKEI,V.HARMAT,G.NARAY-SZABO,             
REMARK   1  AUTH 2 J.OVADI                                                      
REMARK   1  TITL   CRYSTALLIZATION AND PRELIMINARY DIFFRACTION                  
REMARK   1  TITL 2 ANALYSIS OF CA2+ CALMODULIN-DRUG AND                         
REMARK   1  TITL 3 APOCALMODULIN-DRUG COMPLEXES                                 
REMARK   1  REF    PROTEINS: STRUCT.,FUNCT.,     V.  28   131 1997              
REMARK   1  REF  2 GENET.                                                       
REMARK   1  REFN   ASTM PSFGEY  US ISSN 0887-3585                               
REMARK   1 REFERENCE 3                                                          
REMARK   1  AUTH   M.VANDONSELAAR,R.A.HICKIE,J.W.QUAIL,L.T.J.DELBAERE           
REMARK   1  TITL   TRIFLUOPERAZINE-INDUCED CONFORMATIONAL CHANGE IN CA          
REMARK   1  TITL 2 (2+)-CALMODULIN                                              
REMARK   1  REF    NAT.STRUCT.BIOL.              V.   1   795 1994              
REMARK   1  REFN   ASTM NSBIEW  US ISSN 1072-8368                               
REMARK   1 REFERENCE 4                                                          
REMARK   1  AUTH   W.J.COOK,L.J.WALTER,M.R.WALTER                               
REMARK   1  TITL   DRUG BINDING BY CALMODULIN: CRYSTAL STRUCTURE OF A           
REMARK   1  TITL 2 CALMODULIN-TRIFLUOPERAZINE COMPLEX                           
REMARK   1  REF    BIOCHEMISTRY                  V.  33 15259 1994              
REMARK   1  REFN   ASTM BICHAW  US ISSN 0006-2960                               
REMARK   2                                                                      
REMARK   2 RESOLUTION. 2.64 ANGSTROMS.                                          
REMARK   3                                                                      
REMARK   3 REFINEMENT.                                                          
REMARK   3   PROGRAM     : X-PLOR 3.851                                         
REMARK   3   AUTHORS     : BRUNGER                                              
REMARK   3                                                                      
REMARK   3  DATA USED IN REFINEMENT.                                            
REMARK   3   RESOLUTION RANGE HIGH (ANGSTROMS) : 2.64                           
REMARK   3   RESOLUTION RANGE LOW  (ANGSTROMS) : 24.58                          
REMARK   3   DATA CUTOFF            (SIGMA(F)) : 0                              
REMARK   3   DATA CUTOFF HIGH         (ABS(F)) : 1000000                        
REMARK   3   DATA CUTOFF LOW          (ABS(F)) : 0.001                          
REMARK   3   COMPLETENESS (WORKING+TEST)   (%) : 94.3                           
REMARK   3   NUMBER OF REFLECTIONS             : 4965                           
REMARK   3                                                                      
REMARK   3  FIT TO DATA USED IN REFINEMENT.                                     
REMARK   3   CROSS-VALIDATION METHOD          : THROUGHOUT                      
REMARK   3   FREE R VALUE TEST SET SELECTION  : RANDOM                          
REMARK   3   R VALUE            (WORKING SET) : 0.207                           
REMARK   3   FREE R VALUE                     : 0.301                           
REMARK   3   FREE R VALUE TEST SET SIZE   (%) :  5.1                            
REMARK   3   FREE R VALUE TEST SET COUNT      : 259                             
REMARK   3   ESTIMATED ERROR OF FREE R VALUE  : 0.010                           
REMARK   3                                                                      
REMARK   3  FIT IN THE HIGHEST RESOLUTION BIN.                                  
REMARK   3   TOTAL NUMBER OF BINS USED           : 8                            
REMARK   3   BIN RESOLUTION RANGE HIGH       (A) : 2.64                         
REMARK   3   BIN RESOLUTION RANGE LOW        (A) : 2.76                         
REMARK   3   BIN COMPLETENESS (WORKING+TEST) (%) : 85.3                         
REMARK   3   REFLECTIONS IN BIN    (WORKING SET) : 473                          
REMARK   3   BIN R VALUE           (WORKING SET) : 0.228                        
REMARK   3   BIN FREE R VALUE                    : 0.445                        
REMARK   3   BIN FREE R VALUE TEST SET SIZE  (%) : 5.2                          
REMARK   3   BIN FREE R VALUE TEST SET COUNT     : 30                           
REMARK   3   ESTIMATED ERROR OF BIN FREE R VALUE : 0.085                        
REMARK   3                                                                      
REMARK   3  NUMBER OF NON-HYDROGEN ATOMS USED IN REFINEMENT.                    
REMARK   3   PROTEIN ATOMS            : 1096                                    
REMARK   3   NUCLEIC ACID ATOMS       : 0                                       
REMARK   3   HETEROGEN ATOMS          : 80                                      
REMARK   3   SOLVENT ATOMS            : 0                                       
REMARK   3                                                                      
REMARK   3  B VALUES.                                                           
REMARK   3   FROM WILSON PLOT           (A**2) : 28.4                           
REMARK   3   MEAN B VALUE      (OVERALL, A**2) : 28.0                           
REMARK   3   OVERALL ANISOTROPIC B VALUE.                                       
REMARK   3    B11 (A**2) : -0.676                                               
REMARK   3    B22 (A**2) : -0.676                                               
REMARK   3    B33 (A**2) : -2.985                                               
REMARK   3    B12 (A**2) : -1.466                                               
REMARK   3    B13 (A**2) : 0.000                                                
REMARK   3    B23 (A**2) : 0.000                                                
REMARK   3                                                                      
REMARK   3  ESTIMATED COORDINATE ERROR.                                         
REMARK   3   ESD FROM LUZZATI PLOT        (A) : 0.290                           
REMARK   3   ESD FROM SIGMAA              (A) : 0.246                           
REMARK   3   LOW RESOLUTION CUTOFF        (A) : 2.74                            
REMARK   3                                                                      
REMARK   3  CROSS-VALIDATED ESTIMATED COORDINATE ERROR.                         
REMARK   3   ESD FROM C-V LUZZATI PLOT    (A) : 0.431                           
REMARK   3   ESD FROM C-V SIGMAA          (A) : 0.526                           
REMARK   3                                                                      
REMARK   3  RMS DEVIATIONS FROM IDEAL VALUES.                                   
REMARK   3   BOND LENGTHS                 (A) : 0.006                           
REMARK   3   BOND ANGLES            (DEGREES) : 1.358                           
REMARK   3   DIHEDRAL ANGLES        (DEGREES) : 24.234                          
REMARK   3   IMPROPER ANGLES        (DEGREES) : 0.566                           
REMARK   3                                                                      
REMARK   3  ISOTROPIC THERMAL MODEL : GROUP                                     
REMARK   3                                                                      
REMARK   3  ISOTROPIC THERMAL FACTOR RESTRAINTS.    RMS    SIGMA                
REMARK   3   MAIN-CHAIN BOND              (A**2) : NULL  ; NULL                 
REMARK   3   MAIN-CHAIN ANGLE             (A**2) : NULL  ; NULL                 
REMARK   3   SIDE-CHAIN BOND              (A**2) : NULL  ; NULL                 
REMARK   3   SIDE-CHAIN ANGLE             (A**2) : NULL  ; NULL                 
REMARK   3                                                                      
REMARK   3  NCS MODEL : NULL                                                    
REMARK   3                                                                      
REMARK   3  NCS RESTRAINTS.                         RMS   SIGMA/WEIGHT          
REMARK   3   GROUP  1  POSITIONAL            (A) : NULL  ; NULL                 
REMARK   3   GROUP  1  B-FACTOR           (A**2) : NULL  ; NULL                 
REMARK   3                                                                      
REMARK   3  PARAMETER FILE  1  : PROTEIN_REP.PARAM                              
REMARK   3  PARAMETER FILE  2  : CA.PAR                                         
REMARK   3  PARAMETER FILE  3  : AAA.PAR                                        
REMARK   3  TOPOLOGY FILE  1   : TOPHCSDX.PRO                                   
REMARK   3  TOPOLOGY FILE  2   : CA.TOP                                         
REMARK   3  TOPOLOGY FILE  3   : AAA.TOP                                        
REMARK   3                                                                      
REMARK   3  OTHER REFINEMENT REMARKS: DISORDERED SIDE CHAIN ATOMS OF            
REMARK   3   RESIDUES ARG 74 - THR 79 AND SER 81 OF THE CENTRAL REGION,         
REMARK   3   GLU 6, GLU 83, TRIMETHYL-LYSINE 115, GLU 123 AND GLU 127           
REMARK   3   ARE NOT SEEN IN THE CRYSTAL STRUCTURE, AS WELL AS THE              
REMARK   3   N-TERMINAL ALA 1, ASP 2 AND C-TERMINAL ALA 147, LYS 148            
REMARK   3   RESIDUES.                                                          
REMARK   3   TEMPERATURE FACTORS FOR THE ATOMS IN RESIDUES 75 - 81 ARE          
REMARK   3   UNUSUALLY HIGH, INDICATING FLEXIBILITY IN THIS REGION.             
REMARK   3   THE C-TERMINAL RESIDUES WERE NOT SEEN IN THE DENSITY MAPS          
REMARK   4                                                                      
REMARK   4 1QIV COMPLIES WITH FORMAT V. 2.3, 09-JULY-1998                       
REMARK 100                                                                      
REMARK 100 THIS ENTRY HAS BEEN PROCESSED BY EBI  ON 17-JUN-1999.                
REMARK 100 THE EBI ID CODE IS EBI-2823.                                         
REMARK 200                                                                      
REMARK 200 EXPERIMENTAL DETAILS                                                 
REMARK 200  EXPERIMENT TYPE                : X-RAY DIFFRACTION                  
REMARK 200  DATE OF DATA COLLECTION        : 15-AUG-1997                        
REMARK 200  TEMPERATURE           (KELVIN) :  93                                
REMARK 200  PH                             : 5.0                                
REMARK 200  NUMBER OF CRYSTALS USED        : 1                                  
REMARK 200                                                                      
REMARK 200  SYNCHROTRON              (Y/N) : N                                  
REMARK 200  RADIATION SOURCE               : ROTATING ANODE                     
REMARK 200  BEAMLINE                       : NULL                               
REMARK 200  X-RAY GENERATOR MODEL          : RIGAKU RU200                       
REMARK 200  MONOCHROMATIC OR LAUE    (M/L) : M                                  
REMARK 200  WAVELENGTH OR RANGE        (A) : 1.5418                             
REMARK 200  MONOCHROMATOR                  : GRAPHITE                           
REMARK 200  OPTICS                         : NORMAL FOCUS                       
REMARK 200                                                                      
REMARK 200  DETECTOR TYPE                  : IMAGE PLATE                        
REMARK 200  DETECTOR MANUFACTURER          : MARRESEARCH                        
REMARK 200  INTENSITY-INTEGRATION SOFTWARE : DENZO                              
REMARK 200  DATA SCALING SOFTWARE          : SCALEPACK                          
REMARK 200                                                                      
REMARK 200  NUMBER OF UNIQUE REFLECTIONS   : 4969                               
REMARK 200  RESOLUTION RANGE HIGH      (A) : 2.63                               
REMARK 200  RESOLUTION RANGE LOW       (A) : 24.58                              
REMARK 200  REJECTION CRITERIA  (SIGMA(I)) : 0                                  
REMARK 200                                                                      
REMARK 200 OVERALL.                                                             
REMARK 200  COMPLETENESS FOR RANGE     (%) : 92.7                               
REMARK 200  DATA REDUNDANCY                : 4.3                                
REMARK 200  R MERGE                    (I) : 0.058                              
REMARK 200  R SYM                      (I) : NULL                               
REMARK 200  <I/SIGMA(I)> FOR THE DATA SET  : 20.6                               
REMARK 200                                                                      
REMARK 200 IN THE HIGHEST RESOLUTION SHELL.                                     
REMARK 200  HIGHEST RESOLUTION SHELL, RANGE HIGH (A) : 2.63                     
REMARK 200  HIGHEST RESOLUTION SHELL, RANGE LOW  (A) : 2.72                     
REMARK 200  COMPLETENESS FOR SHELL     (%) : 76.2                               
REMARK 200  DATA REDUNDANCY IN SHELL       : 2.3                                
REMARK 200  R MERGE FOR SHELL          (I) : 0.123                              
REMARK 200  R SYM FOR SHELL            (I) : NULL                               
REMARK 200  <I/SIGMA(I)> FOR SHELL         : 9.0                                
REMARK 200                                                                      
REMARK 200 DIFFRACTION PROTOCOL: SINGLE WAVELENGTH                              
REMARK 200 METHOD USED TO DETERMINE THE STRUCTURE: MOLECULAR REPLACEMENT        
REMARK 200 SOFTWARE USED: AMORE                                                 
REMARK 200 STARTING MODEL: PDB ENTRY 1LIN                                       
REMARK 200                                                                      
REMARK 200 REMARK: NULL                                                         
REMARK 280                                                                      
REMARK 280 CRYSTAL                                                              
REMARK 280 SOLVENT CONTENT, VS  (%): 52                                         
REMARK 280 MATTHEWS COEFFICIENT, VM (ANGSTROMS**3/DA): 2.5                      
REMARK 280                                                                      
REMARK 280 CRYSTALLIZATION CONDITIONS: PROTEIN WAS CRYSTALLIZED BY              
REMARK 280  HANGING DROP TECHNIQUE AT ROOM TEMPERATURE FROM 50 MM PH=5.0        
REMARK 280  SODIUM CACODYLATE/HCL BUFFER, 10 MM MGCL2, 10 MM CACL2,             
REMARK 280  2MM DPD AND 28% PEG 8000. CRYSTAL GROWTH TOOK 2-3 WEEKS.            
REMARK 290                                                                      
REMARK 290 CRYSTALLOGRAPHIC SYMMETRY                                            
REMARK 290 SYMMETRY OPERATORS FOR SPACE GROUP:  P 32 2 1                        
REMARK 290                                                                      
REMARK 290      SYMOP   SYMMETRY                                                
REMARK 290     NNNMMM   OPERATOR                                                
REMARK 290       1555   X,Y,Z                                                   
REMARK 290       2555   -Y,X-Y,Z+2/3                                            
REMARK 290       3555   Y-X,-X,Z+1/3                                            
REMARK 290       4555   Y,X,-Z                                                  
REMARK 290       5555   X-Y,-Y,1/3-Z                                            
REMARK 290       6555   -X,Y-X,2/3-Z                                            
REMARK 290                                                                      
REMARK 290     WHERE NNN -> OPERATOR NUMBER                                     
REMARK 290           MMM -> TRANSLATION VECTOR                                  
REMARK 290                                                                      
REMARK 290 CRYSTALLOGRAPHIC SYMMETRY TRANSFORMATIONS                            
REMARK 290 THE FOLLOWING TRANSFORMATIONS OPERATE ON THE ATOM/HETATM             
REMARK 290 RECORDS IN THIS ENTRY TO PRODUCE CRYSTALLOGRAPHICALLY                
REMARK 290 RELATED MOLECULES.                                                   
REMARK 290   SMTRY1   1  1.000000  0.000000  0.000000        0.00000            
REMARK 290   SMTRY2   1  0.000000  1.000000  0.000000        0.00000            
REMARK 290   SMTRY3   1  0.000000  0.000000  1.000000        0.00000            
REMARK 290   SMTRY1   2 -0.500000 -0.866025  0.000000        0.00000            
REMARK 290   SMTRY2   2  0.866025 -0.500000  0.000000        0.00000            
REMARK 290   SMTRY3   2  0.000000  0.000000  1.000000      115.87600            
REMARK 290   SMTRY1   3 -0.500000  0.866025  0.000000        0.00000            
REMARK 290   SMTRY2   3 -0.866025 -0.500000  0.000000        0.00000            
REMARK 290   SMTRY3   3  0.000000  0.000000  1.000000       57.93800            
REMARK 290   SMTRY1   4 -0.500000  0.866025  0.000000        0.00000            
REMARK 290   SMTRY2   4  0.866025  0.500000  0.000000        0.00000            
REMARK 290   SMTRY3   4  0.000000  0.000000 -1.000000        0.00000            
REMARK 290   SMTRY1   5  1.000000  0.000000  0.000000        0.00000            
REMARK 290   SMTRY2   5  0.000000 -1.000000  0.000000        0.00000            
REMARK 290   SMTRY3   5  0.000000  0.000000 -1.000000       57.93800            
REMARK 290   SMTRY1   6 -0.500000 -0.866025  0.000000        0.00000            
REMARK 290   SMTRY2   6 -0.866025  0.500000  0.000000        0.00000            
REMARK 290   SMTRY3   6  0.000000  0.000000 -1.000000      115.87600            
REMARK 290                                                                      
REMARK 290 REMARK: NULL                                                         
REMARK 300                                                                      
REMARK 300 BIOLOGICAL UNIT: MONOMER                                             
REMARK 465                                                                      
REMARK 465 MISSING RESIDUES                                                     
REMARK 465 THE FOLLOWING RESIDUES WERE NOT LOCATED IN THE                       
REMARK 465 EXPERIMENT. (M=MODEL NUMBER; RES=RESIDUE NAME; C=CHAIN               
REMARK 465 IDENTIFIER; SSSEQ=SEQUENCE NUMBER; I=INSERTION CODE):                
REMARK 465                                                                      
REMARK 465   M RES C SSSEQI                                                     
REMARK 465     ALA A     1                                                      
REMARK 465     ASP A     2                                                      
REMARK 465     ALA A   147                                                      
REMARK 465     LYS A   148                                                      
REMARK 470                                                                      
REMARK 470 MISSING ATOM                                                         
REMARK 470 THE FOLLOWING RESIDUES HAVE MISSING ATOMS (M=MODEL NUMBER;           
REMARK 470 RES=RESIDUE NAME; C=CHAIN IDENTIFIER; SSEQ=SEQUENCE NUMBER;          
REMARK 470 I=INSERTION CODE):                                                   
REMARK 470   M RES CSSEQI  ATOMS                                                
REMARK 470     GLU A   6    CG   CD   OE1  OE2                                  
REMARK 470     ARG A  74    CG   CD   NE   CZ   NH1  NH2                        
REMARK 470     LYS A  75    CG   CD   CE   NZ                                   
REMARK 470     MET A  76    CG   SD   CE                                        
REMARK 470     LYS A  77    CG   CD   CE   NZ                                   
REMARK 470     ASP A  78    CG   OD1  OD2                                       
REMARK 470     THR A  79    CB   OG1  CG2                                       
REMARK 470     SER A  81    OG                                                  
REMARK 470     GLU A  83    CD   OE1  OE2                                       
REMARK 470     LYS A 115    CG   CD   CE   NZ                                   
REMARK 470     GLU A 123    CG   CD   OE1  OE2                                  
REMARK 470     GLU A 127    CD   OE1  OE2                                       
REMARK 800                                                                      
REMARK 800 SITE                                                                 
REMARK 800 SITE_IDENTIFIER: CA1                                                 
REMARK 800 SITE_DESCRIPTION: CALCIUM BINDING SITE                               
REMARK 800                                                                      
REMARK 800 SITE_IDENTIFIER: CA2                                                 
REMARK 800 SITE_DESCRIPTION: CALCIUM BINDING SITE                               
REMARK 800                                                                      
REMARK 800 SITE_IDENTIFIER: CA3                                                 
REMARK 800 SITE_DESCRIPTION: CALCIUM BINDING SITE                               
REMARK 800                                                                      
REMARK 800 SITE_IDENTIFIER: CA4                                                 
REMARK 800 SITE_DESCRIPTION: CALCIUM BINDING SITE                               
REMARK 800                                                                      
REMARK 900                                                                      
REMARK 900 RELATED ENTRIES                                                      
REMARK 900 RELATED ID: 1LIN   RELATED DB: PDB                                   
REMARK 900 RELATED ID: 1QIW   RELATED DB: PDB                                   
REMARK 900                                                                      
DBREF  1QIV A    1   148  SWS    P02593   CALM_HUMAN       1    148             
SEQRES   1 A  148  ALA ASP GLN LEU THR GLU GLU GLN ILE ALA GLU PHE LYS          
SEQRES   2 A  148  GLU ALA PHE SER LEU PHE ASP LYS ASP GLY ASP GLY THR          
SEQRES   3 A  148  ILE THR THR LYS GLU LEU GLY THR VAL MET ARG SER LEU          
SEQRES   4 A  148  GLY GLN ASN PRO THR GLU ALA GLU LEU GLN ASP MET ILE          
SEQRES   5 A  148  ASN GLU VAL ASP ALA ASP GLY ASN GLY THR ILE ASP PHE          
SEQRES   6 A  148  PRO GLU PHE LEU THR MET MET ALA ARG LYS MET LYS ASP          
SEQRES   7 A  148  THR ASP SER GLU GLU GLU ILE ARG GLU ALA PHE ARG VAL          
SEQRES   8 A  148  PHE ASP LYS ASP GLY ASN GLY TYR ILE SER ALA ALA GLU          
SEQRES   9 A  148  LEU ARG HIS VAL MET THR ASN LEU GLY GLU LYS LEU THR          
SEQRES  10 A  148  ASP GLU GLU VAL ASP GLU MET ILE ARG GLU ALA ASP ILE          
SEQRES  11 A  148  ASP GLY ASP GLY GLN VAL ASN TYR GLU GLU PHE VAL GLN          
SEQRES  12 A  148  MET MET THR ALA LYS                                          
HET     CA  A 149       1                                                       
HET     CA  A 150       1                                                       
HET     CA  A 151       1                                                       
HET     CA  A 152       1                                                       
HET    DPD  A 153      38                                                       
HET    DPD  A 154      38                                                       
HETNAM      CA CALCIUM ION                                                      
HETNAM     DPD N-(3,3-DIPHENYLPROPYL)-N'-[1-R-(3,4-BIS-BUTOXYPHENYL)ETHYL]-     
HETNAM   2 DPD PROPYLENEDIAMINE                                                 
FORMUL   2   CA    4(CA1 2+)                                                    
FORMUL   3  DPD    2(C34 H48 N2 O2)                                             
HELIX    1   1 THR A    5  ASP A   20  1                                  16    
HELIX    2   2 THR A   28  LEU A   39  1                                  12    
HELIX    3   3 THR A   44  ASP A   56  1                                  13    
HELIX    4   4 PHE A   65  ARG A   74  1                                  10    
HELIX    5   5 SER A   81  ASP A   93  1                                  13    
HELIX    6   6 SER A  101  LEU A  112  1                                  12    
HELIX    7   7 THR A  117  ASP A  129  1                                  13    
HELIX    8   8 ASN A  137  THR A  146  1                                  10    
SHEET    1   A 2 THR A  26  ILE A  27  0                                        
SHEET    2   A 2 ILE A  63  ASP A  64 -1  O  ILE A  63   N  ILE A  27           
LINK        CA    CA A 149                 O   THR A  26                        
LINK        CA    CA A 149                 OD1 ASP A  20                        
LINK        CA    CA A 149                 OD1 ASP A  22                        
LINK        CA    CA A 149                 OD1 ASP A  24                        
LINK        CA    CA A 149                 OE1 GLU A  31                        
LINK        CA    CA A 149                 OE2 GLU A  31                        
LINK        CA    CA A 150                 O   THR A  62                        
LINK        CA    CA A 150                 OD1 ASN A  60                        
LINK        CA    CA A 150                 OD1 ASP A  56                        
LINK        CA    CA A 150                 OD1 ASP A  58                        
LINK        CA    CA A 150                 OE1 GLU A  67                        
LINK        CA    CA A 150                 OE2 GLU A  67                        
LINK        CA    CA A 151                 O   TYR A  99                        
LINK        CA    CA A 151                 OD1 ASN A  97                        
LINK        CA    CA A 151                 OD1 ASP A  93                        
LINK        CA    CA A 151                 OD1 ASP A  95                        
LINK        CA    CA A 151                 OD2 ASP A  95                        
LINK        CA    CA A 151                 OE1 GLU A 104                        
LINK        CA    CA A 151                 OE2 GLU A 104                        
LINK        CA    CA A 152                 O   GLN A 135                        
LINK        CA    CA A 152                 OD1 ASP A 129                        
LINK        CA    CA A 152                 OD1 ASP A 131                        
LINK        CA    CA A 152                 OD1 ASP A 133                        
LINK        CA    CA A 152                 OE1 GLU A 140                        
LINK        CA    CA A 152                 OE2 GLU A 140                        
SITE     1 CA1  5 ASP A  20  ASP A  22  ASP A  24  THR A  26                    
SITE     2 CA1  5 GLU A  31                                                     
SITE     1 CA2  5 ASP A  56  ASP A  58  ASN A  60  THR A  62                    
SITE     2 CA2  5 GLU A  67                                                     
SITE     1 CA3  5 ASP A  93  ASP A  95  ASN A  97  TYR A  99                    
SITE     2 CA3  5 GLU A 104                                                     
SITE     1 CA4  5 ASP A 129  ASP A 131  ASP A 133  GLN A 135                    
SITE     2 CA4  5 GLU A 140                                                     
CRYST1   40.125   40.125  173.814  90.00  90.00 120.00 P 32 2 1      6          
ORIGX1      1.000000  0.000000  0.000000        0.00000                         
ORIGX2      0.000000  1.000000  0.000000        0.00000                         
ORIGX3      0.000000  0.000000  1.000000        0.00000                         
SCALE1      0.024922  0.014389  0.000000        0.00000                         
SCALE2      0.000000  0.028777  0.000000        0.00000                         
SCALE3      0.000000  0.000000  0.005753        0.00000     
(ATOM LINES ARE NOT SHOWN.)
END